Fasalka daawada 1377049-84-7 Velpatasvir ee Daaweynta Cagaarshowga C
Alaabtamagac | Velpatasvir |
La mid ah | GS 5816;Methyl [(2S)-1-[(2S,5S)-2-[9-[2-[(2S,4S)-1-[(2R)-2-[(methoxycarbonyl)amino]-2-phenylacetyl] -4- (methoxymethyl) pyrrolidin-2-yl] -1H-imidazol-5-yl] -1,11-dihydroisochromeno[4',3':6,7]naphtho[1,2-d]imidazol-2- yl] -5-methylpyrrolidin-1-yl] -3-methyl-1-oxobutan-2-yl]carbamate |
CAS Maya. | 1377049-84-7 |
Muuqashada | Caddaan ilaa budo huruud ah |
Qaanuunka molecular | C49H54N8O8 |
Miisaanka Molecular | 883.00 |
Isticmaalka | Darajada daawada ama ujeedada cilmi baarista |
Baakad | Sida ku cad codsigaaga |
Kaydinta | Ku kaydi weel cidhiidhi ah oo iftiin u adkaysta meel qabow |
Velpatasvir Cas: 1377049-84-7 | ||
Walxaha | Heerka | Natiijooyinka |
Muuqashada | Caddaan ilaa budo huruud ah | budo huruud ah oo khafiif ah |
Aqoonsiga | HPLCIR | U hogaansama |
Walxaha laxidhiidha | Wax kasta oo wasakh kale ah ≤0.5%Wadarta wasakhda ≤1.0% | 0.15%0.87% |
Biyaha (KF) | NMT 3.0% | 2.1% |
Xalalka Haraaga ah | Buuxiyay shuruudaha ICH hadda | U hogaansama |
Hadhaaga dabka | NMT 0.2% | U hogaansama |
Biraha culus | NMT 20ppm | U hogaansama |
Qiimayn ( ku salaysan Anhydrous) | 98.0% ~ 102.0% | 98.9% |
Gabagabo:u hoggaansama heerarka gudaha |
Macluumaadka Shirkadda
√ Waayo-aragnimada buuxda ee lakabka maamulka ee warshadda iyo farsamayaqaannada raacsan; √ Tayada had iyo jeer waa tixgelinteena ugu sareysa, nidaamka QC adag; √ 11 sano oo khibrad u leh kooxda iibka dhoofinta; √ shaybaadhka R&D ee madaxa banaan; √ Laba aqoon-is-weydaarsiyo GMP-dheer oo saxeexan; √ Khayraadka hodanka ah ee warshado badan oo shaqo la'aan ah oo loogu talagalay mashruuc la habeeyey; √ Kooxda shaqada oo hufnaan sare leh oo leh waddo joogto ah.Halkan ku qor fariintaada oo noo soo dir